Drug nameMethyltrienolone
DescriptionA synthetic non-aromatizable androgen and anabolic steroid. It binds strongly to the androgen receptor and has therefore also been used as an affinity label for this receptor in the prostate and in prostatic tumors.
DrugBankPrimary Accession Number: DB02998
DINNot available
TypeExperimental, Small Molecule
IndicationNot available
Mechanism of ActionNot available
AbsorptionNot available
ToxicityNot available
Protein BindingNot available
Interactions
RXListNot available
KEGGdrug: Not available / compound: C14257
PubChemcompound: 261000 / substance: 7847067
PharmGKBNot available
Metabolizing Enzymes
NameGeneEntrezIDUniprotSNP
Target
NameGeneEntrezIDSwissprotSNP
Androgen receptorAR367ANDR_RABITrs55686369 rs35025615 rs9332972 rs9332971 rs9332970 rs9332969 rs9332968 rs5902610 rs3032358 rs1800053 rs6154 rs6153 rs6152
Progesterone receptorPGR5241PRGR_HUMANrs1042839 rs500760 rs1042838 rs36055552 rs35747049 rs35131968 rs34852313 rs11571252 rs11571222 rs11571179 rs11571152 rs11571151 rs11571150 rs11571149 rs11571148 rs11571147 rs11571146 rs11571145 rs11571144 rs11571143 rs10160726 rs10160588 rs3740754 rs3740753 rs2020880 rs2020878 rs2020876 rs2020874 rs1379130
FilesDB02998.mol | pdb_859317425473-0.pdb | sdf_7967642414996-0.sdf |
Smilesisomeric:
C[C@]1(O)CC[C@@H]2[C@@H]3CCC4=CC(=O)CCC4=C3C=C[C@]12C
canonical:
CC1(O)CCC2C3CCC4=CC(=O)CCC4=C3C=CC12C

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